上游原料
1-(bromomethyl)cyclohexane6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-ol2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cycloheptene; cyclohexylmethyl 6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-yl ether2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-one2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-ol5-azido-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-yl cyclohexylmethyl ether; 5-azido-2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cycloheptenetert-butyl 2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-ylcarbamatetert-butyl 3-bromo-2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-ylcarbamate9-[(tert-butoxycarbonyl)amino]-3-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cycloheptene-2-carboxylic acidtert-butyl 3-(aminocarbonyl)-2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-ylcarbamate9-amino-3-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cycloheptene-2-carboxamide9-amino-3-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cycloheptene-2-carboxamidemethyl (2S)-2-(acetamido)-3-(3-formyl-4-hydroxyphenyl)propanoatemethyl (2S)-2-(acetamido)-3-[3-(1,3-dithiolan-2-yl)-4-hydroxyphenyl]propanoatemethyl (2S)-2-(acetamido)-3-(3-(1,3-dithiolan-2-yl)-4-[[(trifluoromethyl)sulfonyl]oxy]phenyl)propanoatemethyl 4-[(2S)-2-(acetamido)-3-methoxy-3-oxopropyl]-2-(1,3-dithiolan-2-yl)benzoate(2S)-2-(acetamido)-3-[3-(1,3-dithiolan-2-yl)-4-(methoxycarbonyl)phenyl]propionic acidmethyl 4-((2S)-2-(acetamido)-3-[[3-(aminocarbonyl)-2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-yl]amino]-3-oxopropyl)-2-(1,3-dithiolan-2-yl)benzoatemethyl 4-((2S)-2-(acetamido)-3-[[3-(aminocarbonyl)-2-(cyclohexylmethoxy)-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-5-yl]amino]-3-oxopropyl)-2-formylbenzoate